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A deep learning model for structure-based bioactivity optimization and its application in the bioactivity optimization of a SARS-CoV-2 main protease inhibitor 期刊论文
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2025, 卷号: 291, 页码: 16
作者:  Yang, Zhenyu;  Wang, Kai;  Zhang, Guo;  Jiang, Yuanyuan;  Zeng, Rui;  Qiao, Jingxin;  Li, Yueyue;  Deng, Xinyue;  Xia, Ziyi;  Yao, Rui;  Zeng, Xiaoxi;  Zhang, Liyun;  Zhao, Yi;  Lei, Jian;  Chen, Runsheng
收藏  |  浏览/下载:0/0  |  提交时间:2025/06/25
Structure-based bioactivity optimization  Deep-learning model  SARS-CoV-2 main protease  Molecular scaffold  Pocket-StrMod  
FastTuning: Enabling Fast and Efficient Hyper-Parameter Tuning With Partitioning and Parallelism of Search Space 期刊论文
IEEE TRANSACTIONS ON PARALLEL AND DISTRIBUTED SYSTEMS, 2024, 卷号: 35, 期号: 7, 页码: 1174-1188
作者:  Li, Xiaqing;  Guo, Qi;  Zhang, Guangyan;  Ye, Siwei;  He, Guanhua;  Yao, Yiheng;  Zhang, Rui;  Hao, Yifan;  Du, Zidong;  Zheng, Weimin
收藏  |  浏览/下载:48/0  |  提交时间:2024/12/06
Deep learning  distributed hyper-parameter tuning (HPT) system  parallel computing  
REACT: Remainder Adaptive Compensation for Domain Adaptive Object Detection 期刊论文
IEEE TRANSACTIONS ON IMAGE PROCESSING, 2024, 卷号: 33, 页码: 3735-3748
作者:  Li, Haochen;  Zhang, Rui;  Yao, Hantao;  Zhang, Xin;  Hao, Yifan;  Song, Xinkai;  Li, Ling
收藏  |  浏览/下载:14/0  |  提交时间:2024/12/06
Unsupervised domain adaptation  domain adaptive object detection  feature extraction  prototypes  
Balanced masking strategy for multi-label image classification 期刊论文
NEUROCOMPUTING, 2023, 卷号: 522, 页码: 64-72
作者:  Yuan, Jin;  Zhang, Yao;  Shi, Zhongchao;  Geng, Xin;  Fan, Jianping;  Rui, Yong
收藏  |  浏览/下载:43/0  |  提交时间:2023/07/12
Multi -label image classification  Data imbalance  Masking strategy  Graph neural network  
香山开源高性能RISC-V处理器设计与实现 期刊论文
计算机研究与发展, 2023, 卷号: 60, 期号: 3, 页码: 476
作者:  王凯帆;  徐易难;  余子濠;  唐丹;  陈国凯;  陈熙;  勾凌睿;  胡轩;  金越;  李乾若;  李昕;  蔺嘉炜;  刘彤;  刘志刚;  王华强;  王诲喆;  张传奇;  张发旺;  张林隽;  张紫飞;  张梓悦;  赵阳洋;  周耀阳;  邹江瑞;  蔡晔;  郇丹丹;  李祖松;  赵继业;  何伟;  孙凝晖;  包云岗
收藏  |  浏览/下载:56/0  |  提交时间:2024/05/20
RISC-V  high performance processor  open source  chip design  agile development  RISC-V  高性能处理器  开源  芯片设计  敏捷开发  
Design of an 8-bit Bit-Parallel RSFQ Microprocessor 期刊论文
IEEE TRANSACTIONS ON APPLIED SUPERCONDUCTIVITY, 2020, 卷号: 30, 期号: 7, 页码: 6
作者:  Qu, Pei-Yao;  Tang, Guang-Ming;  Yang, Jia-Hong;  Ye, Xiao-Chun;  Fan, Dong-Rui;  Zhang, Zhi-Min;  Sun, Ning-Hui
收藏  |  浏览/下载:54/0  |  提交时间:2021/12/01
Digital circuit  rapid single-flux-quantum (RSFQ)  superconducting microprocessor  
Bit-Slice Butterfly Processing Units for 64-Point RSFQ FFT Processors 期刊论文
IEEE TRANSACTIONS ON APPLIED SUPERCONDUCTIVITY, 2020, 卷号: 30, 期号: 1, 页码: 6
作者:  Tang, Guang-Ming;  Qu, Pei-Yao;  Zheng, Xiang-Yu;  Yang, Jia-Hong;  Ye, Xiao-Chun;  Fan, Dong-Rui;  Sun, Ning-Hui
收藏  |  浏览/下载:325/0  |  提交时间:2019/12/10
Butterfly processing unit (BPU)  fast Fourier transform (FFT) processor  rapid single flux quantum (RSFQ)  superconducting integrated circuits  
无线通信中的信噪比估计算法研究 期刊论文
计算机工程与应用, 2020, 卷号: 56.0, 期号: 018, 页码: 82
作者:  刘剑锋;  李瑞华;  刘垚圻;  苏泳涛;  胡金龙
收藏  |  浏览/下载:43/0  |  提交时间:2023/12/04
信噪比估计  无线通信  滤波器  上下采样  
Comprehensive identification of peptides in tandem mass spectra using an efficient open search engine 期刊论文
NATURE BIOTECHNOLOGY, 2018, 卷号: 36, 期号: 11, 页码: 1059-+
作者:  Chi, Hao;  Liu, Chao;  Yang, Hao;  Zeng, Wen-Feng;  Wu, Long;  Zhou, Wen-Jing;  Wang, Rui-Min;  Niu, Xiu-Nan;  Ding, Yue-He;  Zhang, Yao;  Wang, Zhao-Wei;  Chen, Zhen-Lin;  Sun, Rui-Xiang;  Liu, Tao;  Tan, Guang-Ming;  Dong, Meng-Qiu;  Xu, Ping;  Zhang, Pei-Heng;  He, Si-Min
收藏  |  浏览/下载:110/0  |  提交时间:2019/08/16
32-Bit 4 x 4 Bit-Slice RSFQ Matrix Multiplier 期刊论文
IEEE TRANSACTIONS ON APPLIED SUPERCONDUCTIVITY, 2018, 卷号: 28, 期号: 7, 页码: 5
作者:  Tang, Guang-Ming;  Qu, Pei-Yao;  Ye, Xiao-Chun;  Fan, Dong-Rui;  Sun, Ning-Hui
收藏  |  浏览/下载:102/0  |  提交时间:2019/12/10
Hardware algorithm  matrix multiplier  micro-processor  rapid single-flux-quantum (RSFQ)  superconducting integrated circuits